Gerhard F. Ecker

Orcid: 0000-0003-4209-6883

Affiliations:
  • University of Vienna, Department of Pharmaceutical Chemistry, Austria


According to our database1, Gerhard F. Ecker authored at least 28 papers between 2002 and 2022.

Collaborative distances:
  • Dijkstra number2 of five.
  • Erdős number3 of four.

Timeline

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Bibliography

2022
Using Jupyter Notebooks for re-training machine learning models.
J. Cheminformatics, 2022

Off-targetP ML: an open source machine learning framework for off-target panel safety assessment of small molecules.
J. Cheminformatics, 2022

KNIME workflow for retrieving causal drug and protein interactions, building networks, and performing topological enrichment analysis demonstrated by a DILI case study.
J. Cheminformatics, 2022

2020
Image Based Liver Toxicity Prediction.
J. Chem. Inf. Model., 2020

COVER: conformational oversampling as data augmentation for molecules.
J. Cheminformatics, 2020

2019
Predicting Residence Time and Drug Unbinding Pathway through Scaled Molecular Dynamics.
J. Chem. Inf. Model., 2019

Conformational Oversampling as Data Augmentation for Molecules.
Proceedings of the Artificial Neural Networks and Machine Learning - ICANN 2019 - 28th International Conference on Artificial Neural Networks, Munich, Germany, September 17-19, 2019, Proceedings, 2019

2018
SAR-Guided Scoring Function and Mutational Validation Reveal the Binding Mode of CGS-8216 at the α1+/γ2- Benzodiazepine Site.
J. Chem. Inf. Model., 2018

Comparing the performance of meta-classifiers - a case study on selected imbalanced data sets relevant for prediction of liver toxicity.
J. Comput. Aided Mol. Des., 2018

2017
Predicting Drug-Induced Cholestasis with the Help of Hepatic Transporters - An <i>in Silico</i> Modeling Approach.
J. Chem. Inf. Model., 2017

Structure based classification for bile salt export pump (BSEP) inhibitors using comparative structural modeling of human BSEP.
J. Comput. Aided Mol. Des., 2017

Empowering pharmacoinformatics by linked life science data.
J. Comput. Aided Mol. Des., 2017

2016
Selectivity profiling of BCRP versus P-gp inhibition: from automated collection of polypharmacology data to multi-label learning.
J. Cheminformatics, 2016

2015
Refinement of the Central Steps of Substrate Transport by the Aspartate Transporter GltPh: Elucidating the Role of the Na2 Sodium Binding Site.
PLoS Comput. Biol., 2015

2014
Ligand and Structure-Based Classification Models for Prediction of P-Glycoprotein Inhibitors.
J. Chem. Inf. Model., 2014

Applicability Domain Analysis (ADAN): A Robust Method for Assessing the Reliability of Drug Property Predictions.
J. Chem. Inf. Model., 2014

2013
Mutational Analysis of the High-Affinity Zinc Binding Site Validates a Refined Human Dopamine Transporter Homology Model.
PLoS Comput. Biol., 2013

Pairwise structural comparison of tiagabine analogs gives new insights into their protein binding modes.
J. Cheminformatics, 2013

2D- and 3D-QSAR studies of a series of benzopyranes and benzopyrano[3, 4b][1, 4]-oxazines as inhibitors of the multidrug transporter P-glycoprotein.
J. Comput. Aided Mol. Des., 2013

2012
Insights into binding events of GABA- and Tiagabine- analogues in the Gamma-Aminobutyric Acid Transporter 1 by means of Molecular Modelling.
J. Cheminformatics, 2012

A computational model for predicting the transport of compounds by ABCC2.
J. Cheminformatics, 2012

2011
Exhaustive Sampling of Docking Poses Reveals Binding Hypotheses for Propafenone Type Inhibitors of P-Glycoprotein.
PLoS Comput. Biol., 2011

2008
On the Relationship Between Feature Selection and Classification Accuracy.
Proceedings of the Third Workshop on New Challenges for Feature Selection in Data Mining and Knowledge Discovery, 2008

2005
Similarity-based descriptors (SIBAR) - A tool for safe exchange of chemical information?
J. Comput. Aided Mol. Des., 2005

2004
Insights into Phenylalanine Derivatives Recognition of VLA-4 Integrin: From a Pharmacophoric Study to 3D-QSAR and Molecular Docking Analyses.
J. Chem. Inf. Model., 2004

Topological Distance Based 3D Descriptors for Use in QSAR and Diversity Analysis.
J. Chem. Inf. Model., 2004

2003
MCASE study of the multidrug resistance reversal activity of propafenone analogs.
J. Comput. Aided Mol. Des., 2003

2002
Similarity based SAR (SIBAR) as tool for early ADME profiling.
J. Comput. Aided Mol. Des., 2002


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